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Carfilzomib (CAS# 868540-17-4)

Ipropati yeMichiza:

Ifomula yeemolekyuli I-C40H57N5O7
IMisa yeMolar 719.92
Ukuxinana 1.161
Indawo yokunyibilika 204 – 208°C
Indawo yeBoling 975.6±65.0 °C(Kuqikelelwe)
Indawo yokuflasha 543.8℃
Ukunyibilika I-Soluble kwi-DMSO (ukuya kwi-80 mg / ml) okanye kwi-Ethanol (ukuya kwi-25 mg / ml).
Uxinzelelo loMphunga 0mmHg ku-25°C
Imbonakalo eqinileyo
Umbala Mhlophe
pKa 13.17±0.46(Kuxelwe kwangaphambili)
Imeko yoGcino -20 °
Uzinzo Izinzile unyaka om-1 ukusuka kumhla wokuthenga njengoko kunikezelwe. Izisombululo kwi-DMSO okanye i-ethanol inokugcinwa kwi--20 ° ukuya kwi-1 iveki.
Refractive Index 1.551
Sebenzisa I-proteasomel inhibitors, i-analogues ye-epoxomicin

Iinkcukacha zeMveliso

Iithegi zeMveliso

Ikhowudi ye-HS 29337900

 

Intshayelelo

I-Carfilzomib (PR-171) i-proteasome inhibitor engenakuguquleka kunye ne-IC50


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